SCHEMBL22014427

SCHEMBL22014427

C=CCc1c(C(C)C)cc(F)cc1C(C)C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.32
GABRA1 P14867 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24785011 0.82 GCGR (0.33) GCGRGABRA1GABRG2GABRB3
SCHEMBL22010373 0.81
SCHEMBL28799188 0.80 GABRA1 (0.47) GABRA1POLB
SCHEMBL9804429 0.80 CA1 (0.35) GABRA1GABRG2GABRB3
SCHEMBL24783786 0.80 GCGR (0.32) GCGRGABRA1GABRG2GABRB3
SCHEMBL24784393 0.77 GABRA1 (0.33) GABRA1GABRG2GABRB3
SCHEMBL25138979 0.76 KDM4E (0.34)
SCHEMBL8125391 0.75 GABRA1 (0.54) GABRA1GABRG2GABRB3
SCHEMBL25138922 0.74 GCGR (0.38) GCGRGABRA1GABRG2GABRB3
SCHEMBL19508138 0.71 NLRP3 (0.36) GCGRGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed