SCHEMBL22014485

SCHEMBL22014485

O=P(O)(O)CN1CCN(Cc2ccc(-c3ccc(CN4CCN(CP(O)O)CCN(CP(O)O)CC4)cc3)cc2)CCN(CP(O)O)CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.47
HRH4 Q9H3N8 1/20 0.44
FAAH O00519 1/20 0.42
CHKA P35790 1/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 1/20 0.41
LSS P48449 1/20 0.40
RORC P51449 1/20 0.40
MCHR1 Q99705 5/20 0.39
CHRM1 P11229 3/20 0.39
HTR2A P28223 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22014104 0.89 HRH3 (0.56) HRH3HRH4FAAHCHKACYP2D6
SCHEMBL22014097 0.84 HRH3 (0.48) HRH3HRH4
SCHEMBL22014095 0.84 FAAH (0.55) HRH3HRH4FAAHCHKACYP2D6
SCHEMBL22014091 0.77 SIGMAR1 (0.64) FAAH
SCHEMBL22014096 0.72 SIGMAR1 (0.49) CYP2D6
SCHEMBL22014099 0.68 MPO (0.53) FAAH
SCHEMBL23532238 0.68 MAPT (0.52)
SCHEMBL3966649 0.68 MAPT (0.52)
SCHEMBL336769 0.68 MAPT (0.52)
SCHEMBL22355488 0.67 SIGMAR1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102820-A1 COMPOUNDS FOR USE AS IRON (III) MRI CONTRAST AGENTS CONTAINING ANIONIC PENDENTS AND ANCILLARY GROUPS THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2020-05-22 WO disclosed