SCHEMBL22014563

SCHEMBL22014563

CC(C)(O)CNC(=O)c1cnc(N)c(C(=N)N2CCCC2)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.39
ACVR1 Q04771 2/20 0.37
PIK3C3 Q8NEB9 1/20 0.36
NPC1 O15118 1/20 0.35
JAK2 O60674 1/20 0.35
NTRK1 P04629 1/20 0.35
CNR2 P34972 2/20 0.35
CFTR P13569 2/20 0.35
TSHR P16473 1/20 0.34
KIT P10721 1/20 0.34
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
TGFBR1 P36897 1/20 0.34
ACVRL1 P37023 1/20 0.34
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24081071 0.80 PHF13 (0.40) NAMPTACVR1KITBMPR1BBMPR1A
SCHEMBL24081049 0.74 BMPR1B (0.53) ACVR1BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL24080970 0.70 NOS3 (0.42) PIK3C3CNR2
SCHEMBL24081037 0.68 MAPK1 (0.45) NAMPTNPC1CNR2
SCHEMBL17298875 0.66 GABRA5 (0.44) NAMPTCNR2CFTR
SCHEMBL28798721 0.65 PIK3C3 (0.46) ACVR1PIK3C3NPC1BMPR1BBMPR1A
SCHEMBL30908079 0.64 NAMPT (0.51) NAMPT
SCHEMBL12302074 0.63 KDM4E (0.60) NAMPTCNR2
SCHEMBL15262659 0.62 MAPK14 (0.44) NAMPTNPC1CNR2CFTRAR
SCHEMBL20788418 0.62 L3MBTL1 (0.57) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098720-A1 FIVE-AND-SIX-MEMBERED HETEROCYCLIC COMPOUND AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITOR 上海轶诺药业有限公司 2020-05-22 WO disclosed