SCHEMBL22017244

SCHEMBL22017244

C=N/C(=C\C=C(/C)NC(=O)c1ccc(OCCCCl)c(N)c1)CN1CCN(C)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
DRD3 P35462 1/20 0.34
HPGD P15428 1/20 0.34
DRD2 P14416 2/20 0.34
HTR2A P28223 2/20 0.34
HTR1A P08908 1/20 0.34
WNT3A P56704 4/20 0.33
CREBBP Q92793 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTR1B P28222 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22017240 0.70 MAPK7 (0.49) WNT3AEGFRMAPK14KIT
SCHEMBL22017241 0.69 KIT (0.62) EGFRKIT
SCHEMBL22018091 0.67 KIT (0.61) EGFRKIT
SCHEMBL28550947 0.66 WNT3A (0.33) MEN1ALDH1A1KMT2AHPGDWNT3A
SCHEMBL28546729 0.63 SRC (0.33) MEN1ALDH1A1KMT2AHPGDWNT3A
SCHEMBL20033130 0.61 PDE4B (0.44) MEN1ALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL10877787 0.60 HTR1B (0.58) HRH3MEN1ALDH1A1KMT2ADRD3
SCHEMBL22017771 0.59 MAPT (0.47) MEN1KMT2AHTR2ACYP2D6CYP2C19
SCHEMBL2949573 0.58 RAD52 (0.61) MEN1ALDH1A1KMT2ADRD3HPGD
SCHEMBL14452258 0.57 DRD2 (0.48) MEN1KMT2ADRD3DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098710-A1 SUBSTITUTED BIS-ARYL AMIDE COMPOUND AND PREPARATION METHOD AND APPLICATION THEREFOR 中国医学科学院医药生物技术研究所 2020-05-22 WO disclosed