SCHEMBL22017588

SCHEMBL22017588

CCC(=O)Nc1cc(C(=O)Nc2ccc(CN3CC(N(C)C)C3)c(C(F)(F)F)c2)ccc1OCCCCl

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 1/20 0.64
ABL1 P00519 6/20 0.49
BCR P11274 3/20 0.49
HCK P08631 1/20 0.48
GCK P35557 1/20 0.48
NR2C2 P49116 1/20 0.48
BRAF P15056 7/20 0.47
EGFR P00533 5/20 0.47
LYN P07948 3/20 0.46
CSK P41240 2/20 0.46
MAPK14 Q16539 2/20 0.46
RIPK2 O43353 1/20 0.46
LCK P06239 1/20 0.46
FYN P06241 1/20 0.46
RET P07949 1/20 0.46
PDGFRB P09619 1/20 0.46
ARAF P10398 1/20 0.46
NQO2 P16083 1/20 0.46
EPHA2 P29317 1/20 0.46
EPHB2 P29323 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22018092 0.88 BRAF (0.60) ABL1BRAFEGFR
SCHEMBL22018093 0.85 BRAF (0.59) ABL1BRAFEGFR
SCHEMBL22017753 0.85 TMPRSS2 (0.87) TMPRSS2ABL1BCRBRAFEGFR
SCHEMBL22017408 0.80 TMPRSS2 (0.79) TMPRSS2ABL1BCRBRAFEGFR
SCHEMBL22018087 0.78 TMPRSS2 (0.54) TMPRSS2HCKNR2C2BRAFEGFR
SCHEMBL22017772 0.77 BRAF (0.64) ABL1BRAFEGFRMAP3K7MAP4K2
SCHEMBL22017247 0.76 BRAF (0.62) ABL1BRAFEGFR
SCHEMBL22017241 0.75 KIT (0.62) ABL1BRAFEGFRRET
SCHEMBL22017577 0.74 CREBBP (0.49) HCKGCKNR2C2BRAFARAF
SCHEMBL22018091 0.72 KIT (0.61) ABL1BRAFEGFRRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098710-A1 SUBSTITUTED BIS-ARYL AMIDE COMPOUND AND PREPARATION METHOD AND APPLICATION THEREFOR 中国医学科学院医药生物技术研究所 2020-05-22 WO disclosed