SCHEMBL22018087

SCHEMBL22018087

CC1CN(Cc2ccc(NC(=O)c3ccc(OCCCCl)c(N)c3)cc2C(F)(F)F)CC(C)O1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 1/20 0.54
HCK P08631 1/20 0.47
NR2C2 P49116 1/20 0.47
BRAF P15056 5/20 0.46
EGFR P00533 4/20 0.46
KIT P10721 3/20 0.46
MAP3K7 O43318 4/20 0.45
MAP4K2 Q12851 4/20 0.45
HTT P42858 2/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44
RET P07949 1/20 0.44
MAPK14 Q16539 3/20 0.43
MAP3K20 Q9NYL2 1/20 0.43
FES P07332 1/20 0.43
FER P16591 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22017241 0.86 KIT (0.62) BRAFEGFRKITRET
SCHEMBL22018091 0.84 KIT (0.61) BRAFEGFRKITRET
SCHEMBL22017771 0.79 MAPT (0.47) HCKNR2C2BRAFEGFRKIT
SCHEMBL22017588 0.78 TMPRSS2 (0.64) TMPRSS2HCKNR2C2BRAFEGFR
SCHEMBL22017753 0.78 TMPRSS2 (0.87) TMPRSS2BRAFEGFRKITRET
SCHEMBL22018092 0.74 BRAF (0.60) BRAFEGFRKIT
SCHEMBL22017242 0.74 TMPRSS2 (0.65) TMPRSS2BRAFKITHTTRET
SCHEMBL22017401 0.74 TMPRSS2 (0.68) TMPRSS2BRAFEGFRKITRET
SCHEMBL22017245 0.73 KIT (0.65) BRAFEGFRKITRET
SCHEMBL31053460 0.72 RAB9A (0.53) TMPRSS2BRAFKITLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020098710-A1 SUBSTITUTED BIS-ARYL AMIDE COMPOUND AND PREPARATION METHOD AND APPLICATION THEREFOR 中国医学科学院医药生物技术研究所 2020-05-22 WO disclosed