SCHEMBL22019130

SCHEMBL22019130

O=C(c1cccc(C(F)(F)F)c1)c1cnc(N2CCC2c2ccccc2)s1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 4/20 0.42
TRPV1 Q8NER1 1/20 0.42
KMT2A Q03164 1/20 0.41
RBP4 P02753 1/20 0.41
MLYCD O95822 2/20 0.41
SRD5A2 P31213 1/20 0.41
SCD O00767 1/20 0.40
SLC6A9 P48067 1/20 0.40
CNR2 P34972 1/20 0.40
CCR2 P41597 2/20 0.40
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962546 1.00 VNN1 (0.42) VNN1TRPV1KMT2ARBP4MLYCD
SCHEMBL22020044 0.91 VNN1 (0.43) VNN1KMT2AMLYCDCNR2CCR2
SCHEMBL21962852 0.91 VNN1 (0.43) VNN1KMT2AMLYCDCNR2CCR2
SCHEMBL21962600 0.83 HPGD (0.42) VNN1TRPV1KMT2ARBP4SRD5A2
SCHEMBL21962542 0.80 RAF1 (0.48) VNN1MLYCDSCDHPGDKDM4E
SCHEMBL21962451 0.80 MEN1 (0.41) VNN1KMT2ARBP4SRD5A2CNR2
SCHEMBL21962674 0.79 SCD (0.47) VNN1MLYCDSCDHPGDKDM4E
SCHEMBL22020041 0.79 ALDH1A1 (0.47) VNN1KMT2AMLYCDSRD5A2SCD
SCHEMBL21962779 0.79 MLYCD (0.49) KMT2AMLYCDSRD5A2SCDHPGD
SCHEMBL21962568 0.79 LMNA (0.51) KMT2AMLYCDSRD5A2SCDHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102575-A1 HETEROCYCLIC AMINOTHIAZOLES AND USES THEREOF INCEPTION IBD, INC. (US) 2020-05-22 WO disclosed