SCHEMBL22040804

SCHEMBL22040804

CC(C)(C)OC(=O)CN1C(=O)OC2(CC3(CC3)c3cc(N)ccc32)C1O

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.34
PLA2G10 O15496 1/20 0.33
PLA2G5 P39877 1/20 0.33
HDAC6 Q9UBN7 2/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22040148 0.77 NR1H2 (0.35) NR1H2
SCHEMBL22040124 0.70 EP300 (0.43)
SCHEMBL23891703 0.69 NR1H2 (0.40) NR1H2PLA2G10PLA2G5
SCHEMBL22040902 0.67 HDAC6 (0.33) HDAC6
SCHEMBL23891672 0.67 CCKBR (0.34) ALDH1A1
SCHEMBL17605850 0.66 EP300 (0.43) NR1H2
SCHEMBL17605847 0.66 EP300 (0.43) NR1H2
SCHEMBL22040127 0.66 EP300 (0.43) NR1H2
SCHEMBL22039456 0.65 BACE1 (0.38) ALDH1A1
SCHEMBL24349905 0.64 EP300 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020108500-A1 HISTONE ACETYLASE P300 INHIBITOR AND USE THEREOF 成都海创药业有限公司 2020-06-04 WO disclosed