SCHEMBL22048877

SCHEMBL22048877

COc1ccc(CN[C@@H](C)I)c(OC)c1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.65
TAS1R3 Q7RTX0 1/20 0.52
TAS1R1 Q7RTX1 1/20 0.52
TSHR P16473 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
LMNA P02545 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105525 0.87 APLNR (0.69) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL24399602 0.84 APLNR (0.65) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL24999551 0.83 APLNR (0.63) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL19138392 0.81 APLNR (0.61) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL19138442 0.81 APLNR (0.61) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL12261590 0.80 APLNR (0.64) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL783785 0.79 APLNR (1.00) APLNRTSHRHTR2AHTR2CCA12
SCHEMBL19138433 0.79 APLNR (0.58) APLNRTAS1R3TAS1R1TSHRHTR2A
SCHEMBL13402596 0.79 APLNR (0.58) APLNRTAS1R3TAS1R1TSHRLMNA
SCHEMBL20079182 0.79 APLNR (0.67) APLNRTSHRHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020112846-A1 SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF NORTHWESTERN UNIVERSITY (US) 2020-06-04 WO disclosed