SCHEMBL22061328

SCHEMBL22061328

CC(C)Nc1ccc(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 4/20 0.40
TBXA2R P21731 2/20 0.39
CSNK1D P48730 1/20 0.39
CSNK1G2 P78368 1/20 0.39
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
KCNJ8 Q15842 1/20 0.37
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
GAA P10253 2/20 0.36
USP30 Q70CQ3 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP11B2 P19099 2/20 0.35
CYP11B1 P15538 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26026410 0.84 MAP2K1 (0.40) MAP2K1CSNK1DCSNK1G2GAAUSP30
SCHEMBL22060849 0.83 ABCC9 (0.40) MAP2K1TBXA2RCSNK1DCSNK1G2ABCC9
SCHEMBL19698925 0.80 TBXA2R (0.40) TBXA2RCSNK1DABCC9ABCC8KCNJ11
SCHEMBL9232027 0.79 MAP2K1 (0.42) MAP2K1CSNK1DCSNK1G2GAAUSP30
SCHEMBL11200089 0.79 MMP13 (0.46) MAP2K1TBXA2RABCB1GAAUSP30
SCHEMBL11200087 0.79 MMP13 (0.46) MAP2K1TBXA2RABCB1GAAUSP30
SCHEMBL2339309 0.79 KDM4E (0.54) TBXA2RABCC9ABCC8KCNJ11KCNJ8
SCHEMBL2814661 0.79 PDK1 (0.47) ABCC9ABCC8KCNJ11KCNJ8ABCB1
SCHEMBL5652691 0.77 PKM (0.39) MAP2K1CSNK1DCSNK1G2ABCC9ABCC8
SCHEMBL21184436 0.76 TBXA2R (0.40) TBXA2RABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020108538-A1 RORγ INHIBITOR HAVING SULFONYL STRUCTURE 正大天晴药业集团股份有限公司 2020-06-04 WO disclosed