SCHEMBL22079235

SCHEMBL22079235

C[C@H](N)c1ccc2[nH]ncc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.55
MAPT P10636 3/20 0.55
ROCK1 Q13464 2/20 0.55
KDM4E B2RXH2 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
RAB9A P51151 1/20 0.55
HIF1A Q16665 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
NOS1 P29475 4/20 0.50
METAP2 P50579 1/20 0.50
CSNK2A1 P68400 1/20 0.50
TRPA1 O75762 2/20 0.48
GSK3B P49841 4/20 0.46
CLK1 P49759 2/20 0.46
DYRK3 O43781 1/20 0.46
CLK2 P49760 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263567 1.00 ROCK2 (0.55) ROCK2MAPTROCK1KDM4EMEN1
SCHEMBL1754871 1.00 ROCK2 (0.55) ROCK2MAPTROCK1KDM4EMEN1
Hydrochloric Acid SCHEMBL28598925 0.98 ROCK2 (0.53) ROCK2MAPTROCK1KDM4EMEN1
Hydrochloric Acid SCHEMBL28598924 0.98 ROCK2 (0.53) ROCK2MAPTROCK1KDM4EMEN1
Hydrochloric Acid SCHEMBL1210017 0.98 ROCK2 (0.53) ROCK2MAPTROCK1KDM4EMEN1
Hydrochloric Acid SCHEMBL1210209 0.98 ROCK2 (0.53) ROCK2MAPTROCK1KDM4EMEN1
Hydrochloric Acid SCHEMBL29915566 0.98 ROCK2 (0.53) ROCK2MAPTROCK1KDM4EMEN1
SCHEMBL18559548 0.86 MAPT (0.55) ROCK2MAPTROCK1KDM4EMEN1
SCHEMBL84462 0.85 TRPA1 (0.54) ROCK2MAPTROCK1KDM4EMEN1
SCHEMBL20841219 0.82 NOS1 (0.55) ROCK2MAPTROCK1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020114949-A1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-06-11 WO disclosed