SCHEMBL22101709

SCHEMBL22101709

CCc1nc2c(F)cc(C)cn2c(=O)c1F

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
AKT3 Q9Y243 1/20 0.31
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 3/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
PKM P14618 1/20 0.31
TSHR P16473 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101422 0.84 MAOB (0.32) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL22101435 0.84 TSHR (0.30) KDM4EALDH1A1HPGDHSD17B10TSHR
SCHEMBL22101184 0.83 CRHR1 (0.31) GRIN1GRIN2AALDH1A1LMNA
SCHEMBL22393763 0.82
SCHEMBL22101706 0.79 HTR1A (0.32) RXFP1LMNA
SCHEMBL22101905 0.79 PDE2A (0.31) KDM4EALDH1A1HSD17B10TSHRRXFP1
SCHEMBL22101725 0.78 GRIN1 (0.40) GRIN1GRIN2AKDM4EALDH1A1HPGD
SCHEMBL23099580 0.77 NPC1 (0.33) ALDH1A1HPGDPKMRXFP1LMNA
SCHEMBL19189767 0.77 ENPP2 (0.30)
SCHEMBL22101707 0.77 ALDH1A1 (0.32) KDM4EALDH1A1HPGDHSD17B10RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed