SCHEMBL22101536

SCHEMBL22101536

Cc1cc(F)c2nc(OCCO)cc(=O)n2c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.38
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.34
IKBKB O14920 1/20 0.33
P2RX7 Q99572 3/20 0.33
POLB P06746 3/20 0.33
MAPT P10636 3/20 0.32
LMNA P02545 2/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TP53 P04637 3/20 0.31
HTT P42858 1/20 0.30
LTB4R Q15722 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22101539 0.87 FFAR4 (0.35) RXFP1POLBMAPTKDM4ENPC1
SCHEMBL22101541 0.85 MAPT (0.35) RXFP1POLBMAPTLMNAKDM4E
SCHEMBL22393587 0.84 THRB (0.33) THRBKMT2AMAPTTP53LTB4R
SCHEMBL22101540 0.81 CYP2C9 (0.35) RXFP1LMNAKDM4EALDH1A1RAB9A
SCHEMBL22101706 0.78 HTR1A (0.32) THRBKMT2ARXFP1P2RX7MAPT
SCHEMBL22101472 0.73 FFAR4 (0.32) ALDH1A1
SCHEMBL22101725 0.72 GRIN1 (0.40) THRBRXFP1POLBMAPTKDM4E
SCHEMBL22393591 0.72 MAPT (0.33) MAPTTP53
SCHEMBL22101868 0.71 KDM4E (0.35) RXFP1MAPTKDM4ESMN1; SMN2
SCHEMBL22101522 0.70 PIK3CB (0.37) PIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed