SCHEMBL22123760

SCHEMBL22123760

NCC(=O)NCC(O)CN

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.42
GABRR1 P24046 3/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADRA1A P35348 1/20 0.37
GABBR2 O75899 1/20 0.32
GABBR1 Q9UBS5 1/20 0.32
TERT O14746 1/20 0.32
GBA1 P04062 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
BCHE P06276 1/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12214451 0.84 MMP2 (0.41) MMP2GABRR1LMNACYP1A2TSHR
SCHEMBL22123634 0.82 MMP2 (0.46) MMP2GABRR1LMNATSHRCYP2C19
SCHEMBL24462473 0.79 CTSD (0.45) GABRR1LMNA
SCHEMBL18342160 0.78
SCHEMBL30171822 0.78
SCHEMBL16197768 0.78
SCHEMBL3180096 0.78
SCHEMBL15833979 0.77 LMNA (0.36) GABRR1LMNACYP1A2TSHRCYP2C19
SCHEMBL16985031 0.77 GABRR1 (0.34) MMP2GABRR1LMNA
SCHEMBL22814737 0.77 ALDH1A1 (0.39) MMP2GABRR1LMNAGABBR2GABBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3898631-A1 NOVEL IMIDAZOPYRAZINE DERIVATIVES AS ANTIBACTERIALS F. Hoffmann-La Roche AG (CH) 2021-10-27 EP disclosed
CN-113195497-A Novel imidazopyrazine derivatives 豪夫迈·罗氏有限公司 2021-07-30 CN disclosed
WO-2020126953-A1 NOVEL IMIDAZOPYRAZINE DERIVATIVES AS ANTIBACTERIALS F. HOFFMANN-LA ROCHE AG (CH) 2020-06-25 WO disclosed