Calycopterin

Calycopterin

SCHEMBL2214965

COc1c(OC)c(O)c2c(=O)c(OC)c(-c3ccc(O)cc3)oc2c1OC

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.73
MAPT P10636 3/20 0.73
GAA P10253 2/20 0.73
TUBB4A P04350 2/20 0.71
TUBB P07437 2/20 0.71
TUBA3C P0DPH7 2/20 0.71
TUBA1B P68363 2/20 0.71
TUBA4A P68366 2/20 0.71
TUBB4B P68371 2/20 0.71
TUBB3 Q13509 2/20 0.71
TUBB2A Q13885 2/20 0.71
TUBB8 Q3ZCM7 2/20 0.71
TUBA3E Q6PEY2 2/20 0.71
TUBA1A Q71U36 2/20 0.71
TUBA1C Q9BQE3 2/20 0.71
TUBB6 Q9BUF5 2/20 0.71
TUBB2B Q9BVA1 2/20 0.71
TUBB1 Q9H4B7 2/20 0.71
ALDH1A1 P00352 1/20 0.67
ABCB1 P08183 3/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31324031 0.92 ABCB1 (0.63) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL4135376 0.92 ABCB1 (0.67) KDM4EMAPTGAATUBB4ATUBB
5-Hydroxyauranetin SCHEMBL4066374 0.90 MAPT (0.71) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL31558901 0.89 MAPT (0.85) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL4129003 0.89 MAPT (0.85) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL29134048 0.85 MAPT (0.64) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL507435 0.84 MAPT (1.00) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL2216677 0.84 KDM4E (0.70) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL571708 0.84 ABCB1 (0.57) KDM4EMAPTGAATUBB4ATUBB
SCHEMBL31080767 0.83 KDM4E (0.67) KDM4EMAPTGAATUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110177237-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2011-07-21 US claimed
WO-2009115051-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2009-09-24 WO claimed
WO-1996031206-A2 FLAVONES AND COUMARINS AS AGENTS FOR THE TREATMENT OF ATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 1996-10-10 WO claimed
CN-117279936-A Fusion proteins comprising proteins with phase behavior 唐纳森公司 2023-12-22 CN disclosed
CN-110312533-B Prodrugs of cytotoxic active agents having enzymatically cleavable groups 拜耳公司 2023-11-03 CN disclosed
CN-114929218-A Treatment of liver diseases using integrin inhibitor combinations 诺华股份有限公司 2022-08-19 CN disclosed
CN-101536687-B Use of flavones and isoflavone derivatives as anti-biofouling substances and method and coating for preventing fouling by marine organisms UNIV HONG KONG SCIENCE & TECHN 2013-12-18 CN disclosed
US-8557331-B2 Antifouling method and composition using chromen-4-one derivatives THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2013-10-15 US disclosed
US-8557331-B2 Antifouling method and composition using chromen-4-one derivatives THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2013-10-15 US disclosed
US-8557331-B2 Antifouling method and composition using chromen-4-one derivatives THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2013-10-15 US disclosed
US-20110177237-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2011-07-21 US disclosed
US-20110177237-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2011-07-21 US disclosed
US-20110177237-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2011-07-21 US disclosed
WO-2009115051-A1 ANTIFOULING METHOD AND COMPOSITION USING CHROMEN-4-ONE DERIVATIVES THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2009-09-24 WO disclosed
CN-101536687-A Use of flavones and isoflavone derivatives as anti-biofouling substances and method and coating for preventing fouling by marine organisms UNIV HONG KONG SCIENCE & TECHN 2009-09-23 CN disclosed
WO-1996031206-A2 FLAVONES AND COUMARINS AS AGENTS FOR THE TREATMENT OF ATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 1996-10-10 WO disclosed