SCHEMBL22199039

SCHEMBL22199039

Cc1ccc(Oc2ccc(OC(F)(F)F)cc2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.46
SLC6A4 P31645 7/20 0.43
SLC6A2 P23975 5/20 0.43
SLC6A3 Q01959 3/20 0.43
SCN8A Q9UQD0 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.41
HTR2A P28223 1/20 0.40
KCNH2 Q12809 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
HSPB1 P04792 1/20 0.39
AR P10275 4/20 0.38
NPBWR1 P48145 1/20 0.38
MCHR1 Q99705 1/20 0.38
BRAF P15056 1/20 0.38
KDR P35968 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199022 0.86 HSPB1 (0.45) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL22199038 0.85 GPR3 (0.47) GPR3SLC6A4SLC6A2SLC6A3SCN8A
SCHEMBL328380 0.82 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL900955 0.82 PDE2A (0.50) GPR3ACHE
SCHEMBL22199016 0.81 ACHE (0.50) HSPB1ARACHE
SCHEMBL1688869 0.81 PPARD (0.44) GPR3SLC6A4SLC6A2SLC6A3SCN8A
SCHEMBL22185629 0.81 SLC6A4 (0.45) SLC6A4SLC6A2SLC6A3
Methane SCHEMBL24038417 0.80 PDE2A (0.49) GPR3ACHE
SCHEMBL16216739 0.80 TSHR (0.45) SLC6A4SLC6A2SLC6A3HTR2AKCNH2
SCHEMBL22184962 0.80 PDE2A (0.47) SLC6A4SLC6A2SLC6A3HSPB1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed