SCHEMBL22201233

SCHEMBL22201233

N=C(CCCc1cccc(Br)c1)OC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.46
FFAR1 O14842 2/20 0.45
FFAR4 Q5NUL3 2/20 0.45
ESR1 P03372 1/20 0.44
NR3C1 P04150 1/20 0.44
PGR P06401 1/20 0.44
NR3C2 P08235 1/20 0.44
AR P10275 1/20 0.44
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
GLS O94925 1/20 0.42
HCAR2 Q8TDS4 1/20 0.42
NPC1 O15118 1/20 0.40
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
PLAAT3 P53816 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21157247 0.91 FFAR1 (0.50) TAAR1FFAR1FFAR4ESR1NR3C1
SCHEMBL21149844 0.83 HDAC1 (0.58) FFAR1NPC1HDAC3HDAC1HDAC2
SCHEMBL21149328 0.82 PLAAT3 (0.47) TAAR1FFAR1FFAR4NPC1HDAC3
SCHEMBL1445967 0.80 HDAC3 (0.63) TAAR1FFAR1FFAR4ESR1NR3C1
SCHEMBL4686018 0.79 TAAR1 (0.50) TAAR1FFAR1FFAR4ESR1NR3C1
SCHEMBL22201278 0.79 MAPT (0.58) FFAR1NPC1HDAC3HDAC1HDAC2
SCHEMBL22201127 0.77 MAPT (0.61) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL22201222 0.77 CYP1A2 (0.66) FFAR1HCAR2HDAC3HDAC1HDAC2
SCHEMBL4686023 0.77 TAAR1 (0.56) TAAR1FFAR1FFAR4ESR1NR3C1
SCHEMBL30828038 0.77 TAAR1 (0.56) TAAR1FFAR1FFAR4ESR1NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141734-A1 METHOD FOR PREPARING CHIRAL GAMMA-LACTAM COMPOUND AND METAL COMPLEX THEREFOR 기초과학연구원 2020-07-09 WO disclosed