SCHEMBL22229733

SCHEMBL22229733

COCOc1c(-c2cccc(COC)c2)cc2c(c1-c1c3c(cc(-c4cccc(COC)c4)c1OCOC)CCCC3)CCCC2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.37
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
FFAR1 O14842 4/20 0.35
RXRA P19793 3/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
TGFBR1 P36897 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
NLRP3 Q96P20 1/20 0.32
RXRB P28702 3/20 0.32
FYN P06241 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
ERN1 O75460 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22256331 0.82 MEN1 (0.52) CYP11B2BRD4CREBBPFFAR1RXRA
SCHEMBL22256328 0.81 L3MBTL1 (0.30) BRD4CREBBPFFAR1L3MBTL1
SCHEMBL22229722 0.76 GPR84 (0.42) CYP11B2BRD4CREBBPFFAR1RXRA
SCHEMBL22229757 0.75 SLC6A2 (0.36) MEN1KMT2ADRD2DRD1ERN1
SCHEMBL22229732 0.75 MEN1 (0.46) MEN1KMT2A
SCHEMBL22229815 0.75 GPR84 (0.37) BRD4CREBBPFFAR1TGFBR1FYN
SCHEMBL22256340 0.73 MEN1 (0.34) MEN1KMT2A
SCHEMBL22229675 0.70 ALDH1A1 (0.33) MEN1KMT2A
SCHEMBL21615685 0.70 PDE4B (0.45) MEN1KMT2A
SCHEMBL22229659 0.69 DHFR (0.39) MEN1KMT2ADRD2DRD1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11664093-B2 Extrapolative prediction of enantioselectivity enabled by computer-driven workflow, new molecular representations and machine learning THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-30 US disclosed
US-11664093-B2 Extrapolative prediction of enantioselectivity enabled by computer-driven workflow, new molecular representations and machine learning THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-30 US disclosed
US-11664093-B2 Extrapolative prediction of enantioselectivity enabled by computer-driven workflow, new molecular representations and machine learning THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-30 US disclosed
US-20200234798-A1 EXTRAPOLATIVE PREDICTION OF ENANTIOSELECTIVITY ENABLED BY COMPUTER-DRIVEN WORKFLOW, NEW MOLECULAR REPRESENTATIONS AND MACHINE LEARNING THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2020-07-23 US disclosed