SCHEMBL22239461

SCHEMBL22239461

CCOC(=O)N1CCCC(c2cc(Cl)nc(Cl)n2)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
HPGD P15428 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 3/20 0.41
GLA P06280 1/20 0.41
RECQL P46063 1/20 0.41
PROKR1 Q8TCW9 2/20 0.41
TSHR P16473 1/20 0.40
KMT2A Q03164 2/20 0.40
MAP3K12 Q12852 1/20 0.40
MEN1 O00255 1/20 0.40
PDE4B Q07343 1/20 0.40
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
POLB P06746 1/20 0.39
CNR1 P21554 2/20 0.39
CNR2 P34972 2/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16220115 0.85 TRPV3 (0.46) ALDH1A1KDM4EHPGDNPSR1HSD17B10
SCHEMBL22123225 0.84 MAP3K12 (0.45) PROKR1MAP3K12
SCHEMBL16220250 0.79 KDM4E (0.46) ALDH1A1KDM4EHPGDNPSR1HSD17B10
SCHEMBL16210779 0.77 TRPV3 (0.46) ALDH1A1KDM4EHPGDHSD17B10GLA
SCHEMBL16211905 0.76 SPR (0.37) MAP3K12RAB9A
SCHEMBL16211959 0.75 MAP3K12 (0.48) PROKR1MAP3K12
SCHEMBL2881051 0.74 JAK2 (0.47) MAP3K12PDE4BRAB9A
SCHEMBL22239462 0.73 PDE4B (0.33) PROKR1MAP3K12PDE4B
SCHEMBL8239996 0.73 POLB (0.40) KDM4EHSD17B10PROKR1KMT2AMAP3K12
SCHEMBL25087319 0.72 MAP3K12 (0.44) PROKR1MAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991977-B1 C-LINKED HETEROCYCLOALKYL SUBSTITUTED PYRIMIDINES AND THEIR USES HOFFMANN LA ROCHE (CH) 2020-07-22 EP disclosed