SCHEMBL22239687

SCHEMBL22239687

Nc1cc(C#CCCOC2(O)CCCCC2)ccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.36
HRH3 Q9Y5N1 1/20 0.32
PAK4 O96013 1/20 0.32
PAK1 Q13153 1/20 0.32
PAK2 Q13177 1/20 0.32
PKN1 Q16512 1/20 0.32
PAK6 Q9NQU5 1/20 0.32
PAK5 Q9P286 1/20 0.32
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
GABRA4 P48169 1/20 0.31
GABRE P78334 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22239573 0.73 QPCT (0.41) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL20385718 0.67 NOS3 (0.43) ASIC3NOS3NOS1NOS2
SCHEMBL18568712 0.66 NOS3 (0.48) ASIC3GABRPGABRDGABRA1GABRB1
SCHEMBL17770071 0.61 HTR1A (0.33) CDC7DBF4
SCHEMBL17770068 0.61 HTR1A (0.33) CDC7DBF4
SCHEMBL28584959 0.59 TSHR (0.30) TSHR
SCHEMBL3498257 0.59 ASIC3 (0.54) ASIC3GABRPGABRDGABRA1GABRB1
SCHEMBL26081246 0.59 TSHR (0.41) USP2TSHR
SCHEMBL26081240 0.59 NOS3 (0.47) HRH3GABRPGABRDGABRA1GABRB1
SCHEMBL2879167 0.58 P2RX7 (0.47) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3221317-B1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2020-07-22 EP disclosed