SCHEMBL2224650

SCHEMBL2224650

COc1cccc(Oc2ncc3nc(-c4cc(C)c([O])c(C)c4)oc3n2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.58
ALDH1A1 P00352 10/20 0.41
HPGD P15428 6/20 0.41
HSD17B10 Q99714 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 2/20 0.41
TP53 P04637 2/20 0.41
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GLA P06280 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KMT2A Q03164 2/20 0.40
F2 P00734 1/20 0.40
USP2 O75604 9/20 0.39
CYP1A2 P05177 9/20 0.39
CYP3A4 P08684 9/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2223355 0.88 S1PR1 (0.73) S1PR1ALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2228933 0.88 S1PR1 (0.58) S1PR1ALDH1A1HPGDHSD17B10KMT2A
SCHEMBL2226291 0.88 S1PR1 (0.55) S1PR1MAPT
SCHEMBL2224909 0.87 S1PR1 (0.58) S1PR1ALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2269044 0.86 S1PR1 (0.55) S1PR1ALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2224272 0.86 S1PR1 (0.55) S1PR1ALDH1A1KDM4EL3MBTL1RAB9A
SCHEMBL14797011 0.85 S1PR1 (0.82) S1PR1ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL2227168 0.84 S1PR1 (0.52) S1PR1ALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2223341 0.83 S1PR1 (0.54) S1PR1ALDH1A1HPGDHSD17B10TP53
SCHEMBL2223895 0.83 S1PR1 (0.52) S1PR1ALDH1A1HPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523962-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2012-11-21 EP disclosed
WO-2011086079-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed