SCHEMBL2228933

SCHEMBL2228933

Cc1cc(-c2nc3cnc(Oc4cccc(F)c4)nc3o2)cc(C)c1[O]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.58
MAOB P27338 2/20 0.39
CETP P11597 2/20 0.39
CYP1A2 P05177 8/20 0.38
CYP3A4 P08684 7/20 0.38
CYP2C9 P11712 7/20 0.38
ALDH1A1 P00352 6/20 0.38
USP2 O75604 5/20 0.38
HSD17B10 Q99714 5/20 0.38
CASP1 P29466 3/20 0.38
CASP7 P55210 3/20 0.38
MAPK1 P28482 1/20 0.38
TSHR P16473 3/20 0.36
CYP2C19 P33261 2/20 0.36
HIF1A Q16665 1/20 0.36
HPGD P15428 4/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
APP P05067 2/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2222401 0.89 S1PR1 (0.49) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL2224650 0.88 S1PR1 (0.58) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL2224142 0.88 S1PR1 (0.51) S1PR1CETPCYP1A2CYP3A4CYP2C9
SCHEMBL2223355 0.88 S1PR1 (0.73) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL2226291 0.87 S1PR1 (0.55) S1PR1CETPEGFRBTKACACB
SCHEMBL2224272 0.87 S1PR1 (0.55) S1PR1CETPCYP1A2CYP2C9ALDH1A1
SCHEMBL2223895 0.86 S1PR1 (0.52) S1PR1MAOBCYP1A2CYP3A4CYP2C9
SCHEMBL2223341 0.86 S1PR1 (0.54) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL2225909 0.86 S1PR1 (0.54) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1
SCHEMBL2224494 0.86 S1PR1 (0.47) S1PR1CYP1A2CYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523962-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2012-11-21 EP disclosed
WO-2011086079-A1 CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed