SCHEMBL22248674

SCHEMBL22248674

Nc1ccn(-c2ccc(CN3CCC4(CC3)CC(N)C4)cc2)c(=O)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.47
CYP2D6 P10635 5/20 0.36
CYP2C9 P11712 4/20 0.36
CYP3A4 P08684 4/20 0.36
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
HIF1A Q16665 2/20 0.33
HPGD P15428 1/20 0.33
USP2 O75604 1/20 0.32
TSHR P16473 3/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CHRM2 P08172 2/20 0.32
CYP1A2 P05177 1/20 0.32
CHRM3 P20309 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
OPRM1 P35372 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22249159 0.90 ROCK2 (0.46) ROCK2CYP2D6CYP2C9CYP3A4MEN1
SCHEMBL22248935 0.89 ROCK2 (0.42) ROCK2OPRM1SIGMAR1
SCHEMBL22248446 0.87 ROCK2 (0.39) ROCK2SIGMAR1
SCHEMBL22248654 0.85 ROCK2 (0.50) ROCK2ALDH1A1SIGMAR1
SCHEMBL22248651 0.83 ROCK2 (0.46) ROCK2OPRM1SIGMAR1
SCHEMBL22249161 0.83 ROCK2 (0.46) ROCK2
SCHEMBL22254490 0.82 ROCK2 (0.49) ROCK2
SCHEMBL22249178 0.81 CYP2D6 (0.47) ROCK2CYP2D6CYP2C9CYP3A4MEN1
SCHEMBL22248655 0.81 ROCK2 (0.47) ROCK2
SCHEMBL22249164 0.78 ROCK2 (0.47) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150372-A1 ANTIMICROBIAL COMPOUNDS AND METHODS CURZA GLOBAL, LLC (US) 2020-07-23 WO disclosed