SCHEMBL22255804

SCHEMBL22255804

CON(C)C(=O)[C@@H](Cc1ccc2ccccc2c1)NC(=O)OC(C)(C)C

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.63
CTSK P43235 6/20 0.63
CTSB P07858 5/20 0.63
PTPN1 P18031 1/20 0.55
MMP9 P14780 1/20 0.54
MMP8 P22894 1/20 0.54
JAK3 P52333 1/20 0.52
BTK Q06187 1/20 0.52
ACE P12821 2/20 0.47
TACR1 P25103 1/20 0.46
CTSL P07711 3/20 0.46
HDAC8 Q9BY41 1/20 0.46
MME P08473 1/20 0.45
KLK5 Q9Y337 1/20 0.44
PIN1 Q13526 1/20 0.43
PPIA P62937 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5993911 1.00 CTSS (0.63) CTSSCTSKCTSBPTPN1MMP9
SCHEMBL29436793 1.00 CTSS (0.63) CTSSCTSKCTSBPTPN1MMP9
SCHEMBL13680202 0.90 MMP9 (0.59) CTSSCTSKCTSBPTPN1MMP9
SCHEMBL1204211 0.86 JAK3 (0.61) CTSSCTSKCTSBJAK3BTK
SCHEMBL6557659 0.86 JAK3 (0.61) CTSSCTSKCTSBJAK3BTK
SCHEMBL9929886 0.85 CTSS (0.62) CTSSCTSKCTSBPTPN1JAK3
SCHEMBL8185213 0.85 CTSS (0.62) CTSSCTSKCTSBPTPN1JAK3
SCHEMBL5630007 0.85 CTSS (0.69) CTSSCTSKCTSBPTPN1MMP9
SCHEMBL31584535 0.85 CTSS (0.69) CTSSCTSKCTSBPTPN1MMP9
SCHEMBL2348036 0.85 MMP9 (0.59) CTSSCTSKCTSBPTPN1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3911645-B1 5-MEMBERED HETEROARYL COMPOUNDS CONTAINING A HYDROXAMATE MOIETY AND THEIR USE UNIV LILLE (FR) 2022-12-07 EP disclosed
WO-2020148403-A1 5-MEMBERED HETEROARYL COMPOUNDS CONTAINING A HYDROXAMATE MOIETY AND THEIR USE UNIVERSITE DE LILLE (FR) 2020-07-23 WO disclosed