SCHEMBL13680202

SCHEMBL13680202

COC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N(C)OC

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.59
MMP8 P22894 2/20 0.59
TACR1 P25103 1/20 0.50
CTSB P07858 3/20 0.49
CTSS P25774 3/20 0.49
CTSL P07711 2/20 0.49
CTSK P43235 2/20 0.49
PIN1 Q13526 1/20 0.47
MME P08473 7/20 0.46
ACE P12821 5/20 0.46
CPA1 P15085 2/20 0.46
ACE2 Q9BYF1 2/20 0.46
PTPN1 P18031 1/20 0.44
FCER2 P06734 1/20 0.44
F2 P00734 1/20 0.44
PPARG P37231 1/20 0.44
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44
PTPRB P23467 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2348036 0.90 MMP9 (0.59) MMP9MMP8TACR1CTSBCTSS
SCHEMBL29436793 0.90 CTSS (0.63) MMP9MMP8TACR1CTSBCTSS
SCHEMBL22255804 0.90 CTSS (0.63) MMP9MMP8TACR1CTSBCTSS
SCHEMBL5993911 0.90 CTSS (0.63) MMP9MMP8TACR1CTSBCTSS
SCHEMBL9910861 0.87 CASP1 (0.52) MMP9MMP8TACR1CTSBCTSS
SCHEMBL6020550 0.85 MMP9 (0.56) MMP9MMP8TACR1CTSBCTSS
SCHEMBL13323301 0.84 MMP9 (0.48) MMP9MMP8TACR1CTSBCTSS
SCHEMBL757454 0.83 MME (0.62) MMP9MMP8TACR1CTSBCTSS
SCHEMBL2779203 0.83 MME (0.62) MMP9MMP8TACR1CTSBCTSS
SCHEMBL6021440 0.81 CTSB (0.53) MMP9MMP8TACR1CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009105825-A1 3-SUBSTITUTED-1,4-DIAZEPAN-2-ONE MELANOCORTIN-5 RECEPTOR ANTAGONISTS MIMETICA PTY LTD (AU) 2009-09-03 WO disclosed