SCHEMBL2225820

SCHEMBL2225820

O=C(O)c1ccc(CC#CO)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
TSHR P16473 3/20 0.50
TP53 P04637 1/20 0.50
SRD5A2 P31213 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
NR4A1 P22736 1/20 0.43
APEX1 P27695 1/20 0.43
APOBEC3A P31941 1/20 0.43
RECQL P46063 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29003644 0.82 KMT2A (0.57) ALDH1A1KMT2APOLBGAAMAPT
SCHEMBL6538715 0.78 ALDH1A1 (0.56) ALDH1A1TSHRTP53SRD5A2KMT2A
SCHEMBL29003606 0.77 LOXL2 (0.58) ALDH1A1TSHRKMT2AKDM4EMEN1
SCHEMBL211305 0.77 ALDH1A1 (0.54) ALDH1A1TSHRTP53SRD5A2KMT2A
SCHEMBL4141280 0.77 ALDH1A1 (0.54) ALDH1A1TSHRTP53SRD5A2KMT2A
SCHEMBL3633156 0.75 FFAR1 (0.44) ALDH1A1TSHRTP53THRBTDP1
Terephthalic Acid SCHEMBL6664013 0.74 TSHR (0.92) ALDH1A1TSHRTP53SRD5A2SMN1; SMN2
SCHEMBL70166 0.72 TSHR (0.67) ALDH1A1TSHRTP53SRD5A2KMT2A
Terephthalic Acid SCHEMBL4612225 0.72 TSHR (0.67) ALDH1A1TSHRTP53SRD5A2KMT2A
SCHEMBL68390 0.72 SRD5A2 (0.69) ALDH1A1TSHRTP53SRD5A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2521727-A1 NOVEL BENZOIC PYRROLOPYRIDINE DERIVATIVES Laboratoires Fournier S.A. (FR) 2012-11-14 EP disclosed
WO-2011083278-A1 NOVEL BENZOIC PYRROLOPYRIDINE DERIVATIVES LABORATOIRES FOURNIER SA (FR) 2011-07-14 WO disclosed