SCHEMBL22258666

SCHEMBL22258666

CC1OCCN(C(=O)Nc2c[nH]nc2-c2ccccn2)C1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
USP2 O75604 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
EPHX2 P34913 4/20 0.34
KCNH2 Q12809 3/20 0.34
CACNA1C Q13936 2/20 0.34
SMO Q99835 1/20 0.34
CYP3A4 P08684 1/20 0.34
SCN5A Q14524 1/20 0.33
P2RX7 Q99572 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579872 0.73 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10MAPTHPGD
SCHEMBL13314749 0.72 SMN1; SMN2 (0.50) ALDH1A1KDM4EHSD17B10HPGDADORA2A
SCHEMBL22258960 0.71 CYP3A4 (0.41) ALDH1A1KDM4EMAPTHPGDCYP3A4
SCHEMBL3588865 0.70 KMT2A (0.45) ALDH1A1KDM4EMEN1KMT2ARAB9A
SCHEMBL22258773 0.70 RAB9A (0.39) ALDH1A1KDM4EHSD17B10MAPTHPGD
SCHEMBL23719268 0.68 ADORA3 (0.51) MAPTADORA2AADORA1EPHX2TSHR
SCHEMBL13314757 0.68 KMT2A (0.54) ALDH1A1KDM4EEPHX2MEN1KMT2A
SCHEMBL13314755 0.66 JAK2 (0.44) MAPTMEN1KMT2ARAB9A
SCHEMBL13314750 0.66 NPC1 (0.49) ALDH1A1MAPTCYP3A4MEN1KMT2A
SCHEMBL13314759 0.65 MCL1 (0.54) ALDH1A1USP2MAPTALOX15CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed