SCHEMBL22258773

SCHEMBL22258773

C[C@H]1CCOCC(C(=O)Nc2c[nH]nc2-c2ccccn2)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
PIP5K1C O60331 4/20 0.37
PIK3CA P42336 4/20 0.37
MAPK10 P53779 2/20 0.37
PIP5K1B O14986 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK14 Q16539 1/20 0.37
PIP5K1A Q99755 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
TGFBR1 P36897 1/20 0.37
ALDH1A1 P00352 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13314749 0.76 SMN1; SMN2 (0.50) RAB9ASMN1; SMN2KDM4EHSD17B10ADORA2A
SCHEMBL3579872 0.73 ALDH1A1 (0.47) RAB9ASMN1; SMN2KDM4EHSD17B10NPC1
SCHEMBL22258960 0.72 CYP3A4 (0.41) KDM4ELMNAALDH1A1L3MBTL1MAPT
SCHEMBL3588865 0.71 KMT2A (0.45) RAB9ASMN1; SMN2KDM4ENPC1ALDH1A1
SCHEMBL22258666 0.70 SCN9A (0.35) RAB9AKDM4EHSD17B10ADORA2AADORA1
SCHEMBL13314757 0.69 KMT2A (0.54) RAB9ASMN1; SMN2KDM4ENPC1ALDH1A1
SCHEMBL13314770 0.69 NPC1 (0.54) RAB9ASMN1; SMN2KDM4EHSD17B10ADORA2A
SCHEMBL23719268 0.68 ADORA3 (0.51) RAB9ASMN1; SMN2ADORA2AADORA2BADORA1
SCHEMBL13314750 0.67 NPC1 (0.49) RAB9ANPC1ALDH1A1MAPT
SCHEMBL415065 0.67 TGFBR1 (0.70) ADORA2AADORA2BADORA1PIP5K1CPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed