SCHEMBL2226437

SCHEMBL2226437

O=C(OCc1ccccc1)N1CCN2c3cccc4[nH]cc(c34)CC2C1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.63
HTR7 P34969 1/20 0.44
HTR5A P47898 1/20 0.44
HTR6 P50406 1/20 0.44
SIGMAR1 Q99720 3/20 0.42
TMEM97 Q5BJF2 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226501 0.82 DRD2 (0.62) DRD2SIGMAR1
SCHEMBL2229717 0.77 DRD2 (1.00) DRD2
SCHEMBL31134492 0.76 ALDH1A1 (0.51) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL6863952 0.75 JAK2 (0.44) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL2229131 0.74 TMEM97 (0.47) SIGMAR1TMEM97NPC1RAB9ASMN1; SMN2
SCHEMBL25342218 0.74 SMN1; SMN2 (0.49) NPC1RAB9ASMN1; SMN2
SCHEMBL11869851 0.74 TMEM97 (0.47) HTR7HTR5AHTR6SIGMAR1TMEM97
SCHEMBL2227321 0.73 HTR6 (0.57) HTR6
SCHEMBL18159771 0.71 SMN1; SMN2 (0.51) NPC1RAB9ASMN1; SMN2
SCHEMBL18149461 0.71 SMN1; SMN2 (0.51) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088836-A1 NOVEL 4-(ARYL-4-SULFONYL)-6,6a,7,8,9,10-HEXAHYDRO-4H-4,8,10a-TRIAZA-ACEPHENANTHRYLENE AND 3-ARYLSULFONYL-6,6a,7,8,9,10-HEXAHYDRO-3H-3,8,10a-TRIAZA-CYCLOPENTA[C]FLUORENE DERIVATIVES AS SEROTONIN 5-HT6 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed