SCHEMBL2226501

SCHEMBL2226501

CC(C)(C)OC(=O)N1CCN2c3cccc4[nH]cc(c34)CC2C1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.62
SIGMAR1 Q99720 5/20 0.45
USP30 Q70CQ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228708 0.85 DRD2 (0.67) DRD2SIGMAR1
SCHEMBL2226437 0.82 DRD2 (0.63) DRD2SIGMAR1
SCHEMBL24187402 0.81 SIGMAR1 (0.65) SIGMAR1USP30
SCHEMBL2226187 0.77 DRD2 (1.00) DRD2
SCHEMBL24187416 0.76 SCN9A (0.49) SIGMAR1USP30
SCHEMBL5705067 0.75 POLB (0.44)
SCHEMBL24187263 0.75 STS (0.46) SIGMAR1USP30
SCHEMBL24187272 0.73 GPR119 (0.46) SIGMAR1USP30
SCHEMBL5704832 0.73 MAPT (0.46)
SCHEMBL1351241 0.73 SIGMAR1 (0.50) SIGMAR1USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed
WO-2011088836-A1 NOVEL 4-(ARYL-4-SULFONYL)-6,6a,7,8,9,10-HEXAHYDRO-4H-4,8,10a-TRIAZA-ACEPHENANTHRYLENE AND 3-ARYLSULFONYL-6,6a,7,8,9,10-HEXAHYDRO-3H-3,8,10a-TRIAZA-CYCLOPENTA[C]FLUORENE DERIVATIVES AS SEROTONIN 5-HT6 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed
WO-2011088836-A1 NOVEL 4-(ARYL-4-SULFONYL)-6,6a,7,8,9,10-HEXAHYDRO-4H-4,8,10a-TRIAZA-ACEPHENANTHRYLENE AND 3-ARYLSULFONYL-6,6a,7,8,9,10-HEXAHYDRO-3H-3,8,10a-TRIAZA-CYCLOPENTA[C]FLUORENE DERIVATIVES AS SEROTONIN 5-HT6 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed