SCHEMBL22279201

SCHEMBL22279201

O=C(Nc1cc(F)c(F)cc1F)n1ccnc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
CD38 P28907 3/20 0.36
ALDH1A1 P00352 2/20 0.36
PKM P14618 1/20 0.36
TNIK Q9UKE5 1/20 0.35
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
BLM P54132 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12018227 0.75 NOX1 (0.44) CA12CA1CA2CA9ALDH1A1
SCHEMBL25003335 0.74 BLM (0.46) CD38MAPTBLM
SCHEMBL9998918 0.73 HPGDS (0.41) ALDH1A1PKMMAPTHTT
SCHEMBL7119064 0.72 MAPT (0.49) ALDH1A1MAPTHTT
SCHEMBL21988033 0.71 AAK1 (0.43) TNIK
SCHEMBL2469763 0.71 CYP19A1 (0.43) ALDH1A1PKMMAPT
SCHEMBL22094785 0.71 GRM4 (0.54) CD38ALDH1A1BLM
SCHEMBL24001003 0.70 MDM2 (0.52) CD38HTT
Imidazole-1-Carboxylic Acid Phenylamide SCHEMBL10668282 0.69 RAB9A (0.50) ALDH1A1PKMHTT
SCHEMBL10662756 0.69 GAA (0.45) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020151756-A1 STABLE SOLID DISPERSIONS OF B-RAF KINASE DIMER INHIBITOR, METHODS OF PREPARATION, AND USES THEREFOR BEIGENE, LTD. (KY) 2020-07-30 WO disclosed