SCHEMBL22280642

SCHEMBL22280642

CCCC[C@H](CC)c1nc(-c2ccc(O)c(C(F)(F)F)c2)no1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.39
GAA P10253 1/20 0.37
XBP1 P17861 1/20 0.37
ATM Q13315 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SPHK2 Q9NRA0 4/20 0.36
SPHK1 Q9NYA1 2/20 0.36
HDAC4 P56524 3/20 0.36
HDAC6 Q9UBN7 2/20 0.36
BMP1 P13497 2/20 0.35
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
HDAC1 Q13547 1/20 0.35
NPY2R P49146 1/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22280466 0.79 SPHK2 (0.49) S1PR1SPHK2SPHK1
SCHEMBL22280486 0.72 SMPD1 (0.53) S1PR1HDAC6HDAC1
SCHEMBL19430707 0.71 SPHK2 (0.53) S1PR1SPHK2
SCHEMBL17666215 0.68 SPHK2 (0.42) S1PR1SPHK2
SCHEMBL22280483 0.67 HDAC4 (0.47) L3MBTL1HDAC4HDAC6HDAC1
SCHEMBL19430786 0.66 S1PR1 (0.47) S1PR1SPHK2
SCHEMBL19430602 0.66 SPHK2 (0.46) S1PR1SPHK2SPHK1BMP1
SCHEMBL20597746 0.66 S1PR1 (0.71) S1PR1
SCHEMBL22280481 0.66 PPARD (0.47) S1PR1ATMNPSR1L3MBTL1SPHK2
SCHEMBL22280272 0.66 SPHK2 (0.39) S1PR1NPSR1SPHK2SPHK1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020154431-A1 INHIBITORS OF SPINSTER HOMOLOG 2 (SPNS2) FOR USE IN THERAPY LYNCH KEVIN R (US) 2020-07-30 WO disclosed