SCHEMBL2228708

SCHEMBL2228708

O=C(O)N1CCN2c3cccc4[nH]cc(c34)CC2C1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.67
SIGMAR1 Q99720 5/20 0.43
PRKD3 O94806 1/20 0.39
PRKCG P05129 1/20 0.39
PRKCB P05771 1/20 0.39
PRKCA P17252 1/20 0.39
PRKCH P24723 1/20 0.39
PRKCI P41743 1/20 0.39
PRKCE Q02156 1/20 0.39
PRKCQ Q04759 1/20 0.39
PRKCZ Q05513 1/20 0.39
PRKCD Q05655 1/20 0.39
PRKD1 Q15139 1/20 0.39
CXCR3 P49682 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226501 0.85 DRD2 (0.62) DRD2SIGMAR1
SCHEMBL2226437 0.83 DRD2 (0.63) DRD2SIGMAR1
SCHEMBL2226187 0.80 DRD2 (1.00) DRD2
SCHEMBL28961218 0.78 SIGMAR1 (0.63) SIGMAR1
SCHEMBL2228354 0.77 DRD2 (1.00) DRD2PRKD3PRKCGPRKCBPRKCA
SCHEMBL2229717 0.77 DRD2 (1.00) DRD2
SCHEMBL2230504 0.75 DRD2 (1.00) DRD2
SCHEMBL2229736 0.75 DRD2 (1.00) DRD2
SCHEMBL30681700 0.75 DRD2 (0.80) DRD2PRKD3PRKCGPRKCBPRKCA
SCHEMBL2286226 0.74 DRD2 (1.00) DRD2PRKD3PRKCGPRKCBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed