SCHEMBL2229094

SCHEMBL2229094

CC(C)=CCc1cccc(N)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.47
MAOA P21397 2/20 0.47
CYP19A1 P11511 2/20 0.46
GGPS1 O95749 1/20 0.42
CYP3A4 P08684 2/20 0.41
CASP1 P29466 1/20 0.41
RECQL P46063 1/20 0.41
NOS1 P29475 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CA14 Q9ULX7 1/20 0.39
F2 P00734 1/20 0.37
PLG P00747 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1904000 0.86 GGPS1 (0.47) MAOBMAOACYP19A1GGPS1CYP3A4
SCHEMBL27346370 0.81 NOS1 (0.51) GGPS1CYP3A4NOS1ALDH1A1
SCHEMBL27314752 0.78 GGPS1 (0.43) CYP19A1GGPS1ALDH1A1TP53AKR1C3
SCHEMBL8848832 0.78 TAAR1 (0.47) MAOBGGPS1ALDH1A1AKR1C3AKR1C2
SCHEMBL2811400 0.78 PRSS1 (0.44) CYP19A1GGPS1NOS1PRSS1PRSS2
SCHEMBL27454646 0.78 MAOB (0.52) MAOBMAOACYP19A1CYP3A4CASP1
SCHEMBL3800542 0.77 AKR1C3 (0.39) CYP19A1GGPS1NOS1ALDH1A1PRSS1
SCHEMBL13189961 0.77 GGPS1 (0.42) MAOBMAOACYP19A1GGPS1CYP3A4
SCHEMBL9454043 0.77 GGPS1 (0.42) MAOBMAOACYP19A1GGPS1CYP3A4
SCHEMBL28041732 0.77 CYP1A2 (0.44) CYP19A1GGPS1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108047142-A Heteroaryl compound and its purposes 阿维拉制药公司 2018-05-18 CN disclosed
EP-2519235-A1 HETEROARYL COMPOUNDS AND USES THEREOF Avila Therapeutics, Inc. (US) 2012-11-07 EP disclosed
WO-2011090760-A1 HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2011-07-28 WO disclosed