SCHEMBL22301893

SCHEMBL22301893

COc1cc(-c2nc3c(C)ccc(C)c3[nH]2)cc(OC)c1OS(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
PARP1 P09874 4/20 0.41
PARP2 Q9UGN5 3/20 0.40
DHODH Q02127 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMPD3 Q9NY59 2/20 0.39
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
NOX1 Q9Y5S8 1/20 0.38
HPSE Q9Y251 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22291214 0.79 SMPD3 (0.58) SMPD3MGAMGAASIMGAM2
SCHEMBL22301855 0.74 CDK4 (0.56) CDK4CCND1PARP1DHODHLMNA
SCHEMBL22291111 0.72 SMPD3 (0.64) CDK4CCND1PARP1PARP2MAPT
SCHEMBL29580411 0.71 ALDH1A1 (0.58) CDK4CCND1LMNAMAPTHTT
SCHEMBL14771418 0.68 MGAM (0.38) MGAMGAASIMGAM2HPSE
SCHEMBL14421949 0.67 ACHE (0.58) LMNAHTT
SCHEMBL21474636 0.65 MGAM (0.61) MGAMGAASIMGAM2
SCHEMBL2494177 0.64 CASR (0.49) PARP1PARP2MGAMGAASI
SCHEMBL2456957 0.64 CYP1A2 (0.46)
SCHEMBL10508622 0.63 MGAM (0.60) PARP1DHODHLMNAMGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220119374-A1 SMALL MOLECULE NEUTRAL SPHINGOMYELINASE 2 (nSMase2) INHIBITORS THE JOHNS HOPKINS UNIVERSITY 2022-04-21 US disclosed
WO-2020160148-A1 SMALL MOLECULE NEUTRAL SPHINGOMYELINASE 2 (NSMASE2) INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2020-08-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220119374-A1 SMALL MOLECULE NEUTRAL SPHINGOMYELINASE 2 (nSMase2) INHIBITORS SMPD2, SPTLC2, SGMS2 CDK4 3727/4885CCND1 3250/4885PARP1 961/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.