SCHEMBL2231986

SCHEMBL2231986

CCCCOC(=O)/C=C/c1cc(C)c(Oc2ccc(OCc3ccc(C#N)cc3)cn2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
ACACB O00763 1/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
AKR1B10 O60218 1/20 0.34
AKR1B1 P15121 1/20 0.34
DPP4 P27487 1/20 0.34
PTGES O14684 1/20 0.33
ALOX5 P09917 1/20 0.33
PPARG P37231 1/20 0.33
P2RX3 P56373 1/20 0.33
APP P05067 1/20 0.33
SCN7A Q01118 1/20 0.33
KCNH2 Q12809 1/20 0.33
ATM Q13315 1/20 0.33
ALOX5AP P20292 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
PLA2G2D Q9UNK4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231809 0.91 ACACB (0.38) ACACBAKR1B10AKR1B1DPP4PTGES
SCHEMBL13582679 0.89 RAB9A (0.40) RAB9ATDP1ACACBCYP4F2CYP4A11
SCHEMBL13582681 0.89 RAB9A (0.40) RAB9ATDP1ACACBCYP4F2CYP4A11
SCHEMBL2231994 0.83 PSEN1 (0.48) PTGESALOX5PPARG
SCHEMBL2233912 0.82 ACACB (0.41) TDP1ACACBAKR1B10AKR1B1DPP4
SCHEMBL13582608 0.80 RAB9A (0.41) RAB9ATDP1ACACBCYP4F2CYP4A11
SCHEMBL13582606 0.80 RAB9A (0.41) RAB9ATDP1ACACBCYP4F2CYP4A11
SCHEMBL13582482 0.79 PTGER3 (0.41) ACACBPPARGMAOB
SCHEMBL13582479 0.79 PTGER3 (0.41) ACACBPPARGMAOB
SCHEMBL2231990 0.79 RAB9A (0.38) RAB9ATDP1ACACBCYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed