SCHEMBL2231994

SCHEMBL2231994

CCCCC(=Cc1cc(C)c(Oc2ccc(OCc3ccc(C#N)cc3)cn2)cc1Cl)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 16/20 0.48
ALOX5 P09917 15/20 0.48
PPARG P37231 12/20 0.48
PTGES O14684 8/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231815 0.91 PSEN1 (0.51) PSEN1ALOX5PPARGPTGES
SCHEMBL13582679 0.84 RAB9A (0.40) PPARG
SCHEMBL13582681 0.84 RAB9A (0.40) PPARG
SCHEMBL2231990 0.84 RAB9A (0.38) PSEN1ALOX5PPARGPTGES
SCHEMBL2231986 0.83 RAB9A (0.38) ALOX5PPARGPTGES
SCHEMBL2233918 0.82 PSEN1 (0.51) PSEN1ALOX5PPARGPTGES
SCHEMBL13582608 0.76 RAB9A (0.41) PPARG
SCHEMBL13582606 0.76 RAB9A (0.41) PPARG
SCHEMBL2235546 0.75 ALOX5 (0.46) PSEN1ALOX5PPARGPTGES
SCHEMBL2231811 0.74 ACACB (0.39) PSEN1ALOX5PPARGPTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed