SCHEMBL2231990

SCHEMBL2231990

CCCC/C(=C\C(=O)O)c1cc(C)c(Oc2ccc(OCc3ccc(C#N)cc3)cn2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.38
ACACB O00763 3/20 0.36
PSEN1 P49768 6/20 0.36
ALOX5 P09917 5/20 0.36
PTGES O14684 4/20 0.36
PPARG P37231 4/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALKBH1 Q13686 1/20 0.35
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
MAOB P27338 2/20 0.34
ACACA Q13085 2/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231811 0.91 ACACB (0.39) ACACBPSEN1ALOX5PTGESPPARG
SCHEMBL2231994 0.84 PSEN1 (0.48) PSEN1ALOX5PTGESPPARG
SCHEMBL2233914 0.82 ACACB (0.41) ACACBPSEN1ALOX5PTGESPPARG
SCHEMBL13582679 0.80 RAB9A (0.40) RAB9AACACBPPARGCYP4F2CYP4A11
SCHEMBL13582681 0.80 RAB9A (0.40) RAB9AACACBPPARGCYP4F2CYP4A11
SCHEMBL2231986 0.79 RAB9A (0.38) RAB9AACACBALOX5PTGESPPARG
SCHEMBL13582608 0.77 RAB9A (0.41) RAB9AACACBPPARGCYP4F2CYP4A11
SCHEMBL13582606 0.77 RAB9A (0.41) RAB9AACACBPPARGCYP4F2CYP4A11
SCHEMBL2235542 0.75 NR4A2 (0.41) RAB9AACACBALKBH1MAOB
SCHEMBL2231815 0.74 PSEN1 (0.51) PSEN1ALOX5PTGESPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed