SCHEMBL22325530

SCHEMBL22325530

c1ccc(COc2cnc(-n3cncn3)nc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALKBH1 Q13686 16/20 0.56
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
TP53 P04637 2/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
P4HTM Q9NXG6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20590806 0.83 NPC1 (0.54) ALKBH1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL4667925 0.81 RAB9A (0.62) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL30723585 0.79 ALKBH1 (0.50) ALKBH1SMN1; SMN2
SCHEMBL1186530 0.78 NPC1 (0.52) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL875608 0.73 LMNA (0.53) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL15952657 0.71 KIT (0.54) ALKBH1NPC1RAB9ASMN1; SMN2P4HTM
SCHEMBL3235402 0.71 NPC1 (0.72) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL30212486 0.70 KCNH2 (0.47) NPC1RAB9ASMN1; SMN2TP53LMNA
SCHEMBL22325535 0.70 CYP2A6 (0.40) SMN1; SMN2LMNAMAPT
SCHEMBL15953346 0.70 KIT (0.53) ALKBH1NPC1RAB9ASMN1; SMN2P4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020162612-A1 PYRIDINE COMPOUND SUBSTITUTED BY HETEROARYL 大正製薬株式会社 2020-08-13 WO disclosed