SCHEMBL22325979

SCHEMBL22325979

Nc1ccc(Br)c(Oc2ccccc2)c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.42
LTA4H P09960 3/20 0.41
TSHR P16473 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
MAOB P27338 1/20 0.38
KMT2A Q03164 4/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SOS1 Q07889 1/20 0.36
KDM1A O60341 1/20 0.36
MEN1 O00255 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22325766 0.84 MEN1 (0.40) TSHRCA1CA2CA12CA7
SCHEMBL22325738 0.81 MAOA (0.47) MAOALTA4HTSHRMAOBKMT2A
SCHEMBL16738884 0.81 THRA (0.42) MAOALTA4HTSHRCA1CA2
SCHEMBL16738910 0.81 NUDT1 (0.38) MAOALTA4HTSHRCA1CA2
SCHEMBL22326109 0.81 MEN1 (0.37) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL22325783 0.80 L3MBTL1 (0.40) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6048021 0.78 CYP1A2 (0.50) MAOALTA4HTSHRMAOBKMT2A
SCHEMBL28597896 0.78 CYP1A2 (0.46) MAOALTA4HTSHRCA1CA2
SCHEMBL22326024 0.78 MAOB (0.44) MAOALTA4HTSHRCA1CA2
SCHEMBL20535327 0.77 RHEB (0.47) MAOALTA4HTSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020162471-A1 PYRIDONE DERIVATIVE マルホ株式会社 2020-08-13 WO disclosed
WO-2020162471-A1 PYRIDONE DERIVATIVE マルホ株式会社 2020-08-13 WO disclosed