SCHEMBL22337997

SCHEMBL22337997

CCC/C(C)=N/OCC(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.39
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
HMGCR P04035 1/20 0.34
CA12 O43570 3/20 0.33
CA14 Q9ULX7 3/20 0.33
POLB P06746 1/20 0.33
POLA1 P09884 1/20 0.33
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC3 O15379 2/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC2 Q92769 2/20 0.31
HDAC8 Q9BY41 2/20 0.31
HDAC6 Q9UBN7 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980204 0.77 GAA (0.44) TSHRGAAALDH1A1MGAMSI
SCHEMBL14587949 0.73 ALDH1A1 (0.37) TSHRGAAALDH1A1KMT2AHDAC3
SCHEMBL4652664 0.71
SCHEMBL10864918 0.71 TSHR (0.40) TSHRGAAALDH1A1MGAMSI
SCHEMBL10932294 0.71 MGAM (0.38) TSHRGAAMGAMSIMGAM2
SCHEMBL1121924 0.71 GAA (0.38) TSHRGAAALDH1A1MGAMSI
SCHEMBL22337986 0.70 MGAM (0.34) TSHRGAAMGAMSIMGAM2
SCHEMBL19770786 0.69
SCHEMBL212133 0.69
SCHEMBL212132 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10875822-B2 Directed β-C(sp3)#H iodination and arylation of ketones THE SCRIPPS RESEARCH INSTITUTE (US) 2020-12-29 US disclosed
US-20200255363-A1 Directed Beta-C(sp3)–H Iodination and Arylation of Ketones THE SCRIPPS RESEARCH INSTITUTE 2020-08-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200255363-A1 Directed Beta-C(sp3)–H Iodination and Arylation of Ketones BCAT1, AOC3, SPIN3 TSHR 797/4885GAA 3962/4885ALDH1A1 1244/4885
US-10875822-B2 Directed β-C(sp3)#H iodination and arylation of ketones BCAT1, AOC3, SPIN3 TSHR 726/4885GAA 4099/4885ALDH1A1 1290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.