SCHEMBL2233904

SCHEMBL2233904

CC(C)(C)OC(=O)NC(C(=O)O)c1cccc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.50
CTSS P25774 1/20 0.50
CPN1 P15169 1/20 0.43
CPB2 Q96IY4 1/20 0.43
GABRB1 P18505 1/20 0.42
GABRB2 P47870 1/20 0.42
ACE P12821 1/20 0.41
S1PR3 Q99500 2/20 0.41
ATM Q13315 2/20 0.41
KLK5 Q9Y337 1/20 0.41
MAPT P10636 1/20 0.40
PPARA Q07869 2/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9261922 1.00 CTSK (0.50) CTSKCTSSCPN1CPB2GABRB1
SCHEMBL11065297 1.00 CTSK (0.50) CTSKCTSSCPN1CPB2GABRB1
SCHEMBL6546992 0.89 CTSK (0.47) CTSKCTSSCPN1CPB2GABRB1
SCHEMBL10093129 0.88 CTSS (0.46) CTSKCTSSGABRB1GABRB2S1PR3
SCHEMBL3618570 0.88 CTSS (0.46) CTSKCTSSGABRB1GABRB2S1PR3
SCHEMBL27204311 0.85 CTSK (0.51) CTSKCTSSGABRB1GABRB2ACE
SCHEMBL10891091 0.85 CTSK (0.51) CTSKCTSSGABRB1GABRB2ACE
SCHEMBL14161705 0.85 CTSK (0.51) CTSKCTSSGABRB1GABRB2ACE
SCHEMBL31230471 0.85 CTSK (0.51) CTSKCTSSGABRB1GABRB2ACE
SCHEMBL116386 0.84 CTSK (0.66) CTSKCTSSGABRB1GABRB2ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4720058-A2 BIFUNCTIONAL DEGRADERS AND USES THEREOF Casma Therapeutics, Inc. (US) 2026-04-08 EP disclosed
WO-2024249291-A2 BIFUNCTIONAL DEGRADERS AND USES THEREOF CASMA THERAPEUTICS, INC. (US) 2024-12-05 WO disclosed
EP-2349990-B1 ARYL-PHENYL-SULFONAMIDE-PHENYLENE COMPOUNDS AND THEIR USE PIMCO 2664 LTD (GB) 2018-05-02 EP disclosed
US-8207167-B2 Aryl-phenyl-sulfonamide-phenylene compounds and their use PIMCO 2664 LIMITED (GB) 2012-06-26 US disclosed
US-20110190302-A1 Aryl-Phenyl-Sulfonamide-Phenylene Compounds and Their Use PIMCO 2664 LIMITED (GB) 2011-08-04 US disclosed
US-5378838-A FOR USE IN HUMANS MERCK & CO., INC. (US) 1995-01-03 US disclosed
WO-1994015924-A1 CHOLECYSTOKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-07-21 WO disclosed
US-4091227-A ANTIBACTERIAL AGENTS SMITHKLINE CORPORATION (US) 1978-05-23 US disclosed
US-4067977-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1978-01-10 US disclosed
US-4067976-A BACTERICIDES SMITHKLINE CORPORATION (US) 1978-01-10 US disclosed
US-4067978-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1978-01-10 US disclosed
US-4007173-A BACTERICIDE SMITHKLINE CORPORATION (US) 1977-02-08 US disclosed
US-3988451-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-10-26 US disclosed
US-3931160-A BACTERICIDE SMITHKLINE CORPORATION (US) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190302-A1 Aryl-Phenyl-Sulfonamide-Phenylene Compounds and Their Use SOST, PSAP, ARSA CTSK 240/4885CTSS 114/4885CPN1 1609/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.