SCHEMBL22343764

SCHEMBL22343764

Nc1ncnc2c1ncn2[C@@H]1O[C@H](COc2cc(CCC(=O)c3ccccc3C(=O)O)cc(C(F)(F)F)c2)[C@@H](O)[C@H]1O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.54
TRDMT1 O14717 2/20 0.52
NT5E P21589 2/20 0.51
GNMT Q14749 1/20 0.50
TRPM2 O94759 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29702996 0.90 ADORA1 (0.54) ADORA1GNMTTRPM2
SCHEMBL22343533 0.89 GNMT (0.57) ADORA1NT5EGNMTTRPM2
SCHEMBL22343666 0.88 GNMT (0.56) ADORA1NT5EGNMTTRPM2
SCHEMBL22343675 0.87 ADH1A (0.53) ADORA1GNMTTRPM2
SCHEMBL22343765 0.85 BCHE (0.42) ADORA1TRDMT1NT5EGNMT
SCHEMBL22323629 0.84 GNMT (0.56) ADORA1NT5EGNMTTRPM2
SCHEMBL29702967 0.81 ADORA1 (0.52) ADORA1GNMTTRPM2
SCHEMBL22343548 0.81 ADORA1 (0.52) ADORA1GNMTTRPM2
SCHEMBL22343662 0.79 BCHE (0.48) ADORA1NT5EGNMT
SCHEMBL1434032 0.77 ADORA1 (0.72) ADORA1TRPM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020163673-A1 INHIBITORS OF ADENYLATE-FORMING ENZYME MENE MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2020-08-13 WO disclosed