SCHEMBL22357571

SCHEMBL22357571

c1ccc(-c2cc(-c3ccc(-c4ccc5nc6n(-c7ccccc7)c7ccccc7n6c5c4)cc3)nc(-c3ccccc3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.41
MEN1 O00255 7/20 0.41
MAPT P10636 6/20 0.41
HPGD P15428 6/20 0.41
ALDH1A1 P00352 5/20 0.41
NTSR1 P30989 1/20 0.41
ADORA1 P30542 3/20 0.40
ADORA2B P29275 2/20 0.40
KDM4E B2RXH2 3/20 0.37
LMNA P02545 2/20 0.37
GLA P06280 1/20 0.37
AVPR1A P37288 1/20 0.37
ADORA2A P29274 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22357648 1.00 KMT2A (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357664 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357649 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357615 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357568 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL25106483 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357561 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357663 0.95 MEN1 (0.41) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357652 0.94 ADORA2B (0.42) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL22357609 0.93 KMT2A (0.41) KMT2AMEN1MAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-09-28 US disclosed
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-09-28 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
US-20230174560-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-06-08 US disclosed
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-05-25 US disclosed
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-05-25 US disclosed
US-20230069900-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-03-09 US disclosed
US-11552258-B2 Organic light-emitting device comprising emission layer satisfying specific singlet excitation energy level conditions SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-01-10 US disclosed
US-20220149287-A1 ORGANIC LIGHT-EMITTING DEVICE Research & Business Foundation Sungkyunkwan University (KR) 2022-05-12 US disclosed
US-20210284906-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-09-16 US disclosed
US-20200321537-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2020-10-08 US disclosed
US-20200266360-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2020-08-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200266360-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME CCNE2, CRY1, CCNE1 KMT2A 2486/4885MEN1 89/4885MAPT 916/4885
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CYP1A1, CYP2E1, AOX1 KMT2A 1066/4885MEN1 334/4885MAPT 2508/4885
US-20230174560-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CRY1, AOX1, CYP1A1 KMT2A 1345/4885MEN1 318/4885MAPT 2009/4885
US-11552258-B2 Organic light-emitting device comprising emission layer satisfying specific singlet excitation energy level conditions EML4, NES, TBL2 KMT2A 1088/4885MEN1 1181/4885MAPT 141/4885
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE L1CAM, EML4, OR10J3 KMT2A 2016/4885MEN1 2788/4885MAPT 527/4885
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CRY1, AOX1, CYP1A1 KMT2A 1497/4885MEN1 367/4885MAPT 2220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.