SCHEMBL22366372

SCHEMBL22366372

O=C(O)N1CCC[C@H](COCCOCCOCc2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSK P43235 1/20 0.46
CHRNB2 P17787 3/20 0.44
CHRNA4 P43681 3/20 0.44
TEAD3 Q99594 2/20 0.44
CHRNB4 P30926 2/20 0.43
CHRNA3 P32297 2/20 0.43
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
MAOB P27338 1/20 0.42
HSD11B1 P28845 1/20 0.42
AGTR2 P50052 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22319963 1.00 CTSL (0.46) CTSLCTSBCTSKCHRNB2CHRNA4
SCHEMBL22616969 0.92 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNA4
SCHEMBL22616971 0.92 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNA4
SCHEMBL22616980 0.92 CTSL (0.53) CTSLCTSBCTSKCHRNB2CHRNA4
SCHEMBL3356243 0.86 TEAD3 (0.47) CTSKCHRNB2CHRNA4TEAD3HSD11B1
SCHEMBL3356236 0.86 TEAD3 (0.47) CTSKCHRNB2CHRNA4TEAD3HSD11B1
SCHEMBL3356619 0.86 TEAD3 (0.47) CTSKCHRNB2CHRNA4TEAD3HSD11B1
SCHEMBL25383877 0.86 HTR6 (0.50) BCHE
SCHEMBL5237806 0.85 SMN1; SMN2 (0.51) CTSLCTSBCTSKCHRNB2CHRNA4
SCHEMBL5229819 0.81 HTR6 (0.50) BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3700911-A1 NOVEL MACROCYCLIC DERIVATIVES, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Les Laboratoires Servier SAS (FR) 2020-09-02 EP disclosed