SCHEMBL2238044

SCHEMBL2238044

NS(=O)(=O)c1cccc(NS(=O)(=O)c2ccc(Br)cc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.58
CA1 P00915 10/20 0.58
CA9 Q16790 2/20 0.58
CA7 P43166 1/20 0.58
CA14 Q9ULX7 1/20 0.58
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
PGR P06401 1/20 0.47
PTGES2 Q9H7Z7 1/20 0.46
HSD11B1 P28845 1/20 0.46
ITGA1 P56199 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CA4 P22748 1/20 0.44
WDR5 P61964 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2237044 0.80 CA2 (0.75) CA2CA1CA9MEN1KMT2A
SCHEMBL13028571 0.78 CA1 (0.57) CA2CA1CA9CA7CA14
SCHEMBL2236215 0.77 CDK1 (0.53) CA2CA1CA9CA7PTGES2
SCHEMBL2237325 0.75 CA2 (0.47) CA2CA1MEN1KMT2APTGES2
SCHEMBL2308296 0.74 CA2 (0.79) CA2CA1CA9MEN1KMT2A
SCHEMBL13552707 0.73 CES1 (0.57) CA2CA1CA9CA7CA14
SCHEMBL841673 0.73 CA2 (0.51) CA2CA1CA9CA7CA14
Methane SCHEMBL11683447 0.73 MEN1 (0.59) CA2CA1MEN1KMT2APGR
SCHEMBL28513727 0.72 HTR6 (0.55) CA2CA1CA9CA7CA14
SCHEMBL11078586 0.72 CA2 (0.49) CA2CA1CA9CA7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349990-B1 ARYL-PHENYL-SULFONAMIDE-PHENYLENE COMPOUNDS AND THEIR USE PIMCO 2664 LTD (GB) 2018-05-02 EP disclosed
US-8207167-B2 Aryl-phenyl-sulfonamide-phenylene compounds and their use PIMCO 2664 LIMITED (GB) 2012-06-26 US disclosed
US-8207167-B2 Aryl-phenyl-sulfonamide-phenylene compounds and their use PIMCO 2664 LIMITED (GB) 2012-06-26 US disclosed
US-20110190302-A1 Aryl-Phenyl-Sulfonamide-Phenylene Compounds and Their Use PIMCO 2664 LIMITED (GB) 2011-08-04 US disclosed
US-20110190302-A1 Aryl-Phenyl-Sulfonamide-Phenylene Compounds and Their Use PIMCO 2664 LIMITED (GB) 2011-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190302-A1 Aryl-Phenyl-Sulfonamide-Phenylene Compounds and Their Use SOST, PSAP, ARSA CA2 2774/4885CA1 3022/4885CA9 2330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.