SCHEMBL2238698

SCHEMBL2238698

NC(CC(=O)O)NC(=O)c1cscn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
MAP3K5 Q99683 1/20 0.40
HDAC3 O15379 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
PIM1 P11309 1/20 0.35
MCHR1 Q99705 1/20 0.35
GRM4 Q14833 1/20 0.34
GRM5 P41594 1/20 0.34
CTSA P10619 6/20 0.34
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2364022 0.83 KDM4E (0.41) KDM4EMAP3K5HDAC3HDAC1HDAC4
SCHEMBL2240079 0.76 KMT2A (0.48) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL4542700 0.75
SCHEMBL31307605 0.74 KDM4E (0.47) KDM4EMAP3K5HDAC3HDAC1HDAC4
SCHEMBL12411796 0.74 KDM4E (0.50) KDM4EMAP3K5PIM1GRM4GRM5
SCHEMBL1768624 0.73 KDM4E (0.46) KDM4EHDAC3HDAC1
SCHEMBL2238850 0.72 P2RX7 (0.59) KDM4EGRM4GRM5CTSA
SCHEMBL15997875 0.71 KDM4E (0.44) KDM4EMAP3K5HDAC3HDAC1HDAC4
SCHEMBL1768726 0.71 HDAC3 (0.45) KDM4EMAP3K5HDAC3HDAC1HDAC6
SCHEMBL2237622 0.70 HSPA9 (0.46) HDAC3HDAC1GRM5CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531520-A1 TEMPLATE-FIXED PEPTIDOMIMETICS WITH CXCR7 MODULATING ACTIVITY Polyphor AG (CH) 2012-12-12 EP disclosed
WO-2011095607-A1 TEMPLATE-FIXED PEPTIDOMIMETICS WITH CXCR7 MODULATING ACTIVITY POLYPHOR AG (CH) 2011-08-11 WO disclosed