SCHEMBL2240809

SCHEMBL2240809

Cc1ccccc1NS(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.71
KEAP1 Q14145 2/20 0.67
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64
CA9 Q16790 1/20 0.64
TSHR P16473 1/20 0.60
KMT2A Q03164 4/20 0.59
MEN1 O00255 3/20 0.57
LMNA P02545 2/20 0.57
HPGD P15428 1/20 0.57
L3MBTL1 Q9Y468 2/20 0.56
USP2 O75604 1/20 0.56
POLB P06746 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
NOD2 Q9HC29 1/20 0.56
KDM4E B2RXH2 1/20 0.54
PKM P14618 2/20 0.54
GAA P10253 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623054 0.86 ALDH1A1 (0.75) ALDH1A1KEAP1CA1CA2CA9
SCHEMBL834586 0.86 ALDH1A1 (0.75) ALDH1A1KEAP1CA2CA9TSHR
SCHEMBL30102910 0.85 ALDH1A1 (0.74) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL1116405 0.85 ALDH1A1 (0.74) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL23057258 0.84 ALDH1A1 (0.73) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL23555160 0.83 ALDH1A1 (0.71) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL31681420 0.83 ALDH1A1 (0.71) ALDH1A1KEAP1CA2CA9TSHR
SCHEMBL3081594 0.83 ALDH1A1 (0.71) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL1592863 0.83 ALDH1A1 (0.71) ALDH1A1KEAP1TSHRKMT2AMEN1
SCHEMBL13875339 0.83 ALDH1A1 (0.71) ALDH1A1KEAP1TSHRKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242496-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-08-03 US disclosed
US-20230242496-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-08-03 US disclosed
US-8673910-B2 Proteasome inhibitors for selectively inducing apoptosis in cancer cells H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE (US) 2014-03-18 US disclosed
US-8673910-B2 Proteasome inhibitors for selectively inducing apoptosis in cancer cells H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE (US) 2014-03-18 US disclosed
US-8673910-B2 Proteasome inhibitors for selectively inducing apoptosis in cancer cells H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE (US) 2014-03-18 US disclosed
WO-2012142698-A1 ALKYLUREA DERIVATIVES ACTIVE AGAINST CANCER CELLS UNIVERSITE LAVAL (CA) 2012-10-26 WO disclosed
US-20110201609-A1 PROTEASOME INHIBITORS FOR SELECTIVELY INDUCING APOPTOSIS IN CANCER CELLS H. LEE MOFFITT CANCER CENTER & RESEARCH INSTITUTE (US) 2011-08-18 US disclosed
US-20110201609-A1 PROTEASOME INHIBITORS FOR SELECTIVELY INDUCING APOPTOSIS IN CANCER CELLS H. LEE MOFFITT CANCER CENTER & RESEARCH INSTITUTE (US) 2011-08-18 US disclosed
US-20110201609-A1 PROTEASOME INHIBITORS FOR SELECTIVELY INDUCING APOPTOSIS IN CANCER CELLS H. LEE MOFFITT CANCER CENTER & RESEARCH INSTITUTE (US) 2011-08-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242496-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA BCL6, SOX18, BCL3 ALDH1A1 2654/4885KEAP1 463/4885CA1 3919/4885
US-20110201609-A1 PROTEASOME INHIBITORS FOR SELECTIVELY INDUCING APOPTOSIS IN CANCER CELLS PSMB7, PSMD7, PSMB6 ALDH1A1 4279/4885KEAP1 332/4885CA1 1931/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.