SCHEMBL22453086

SCHEMBL22453086

Cc1cc(N(C)c2ccc(C3CCCCC3)cc2Cl)ccc1Nc1cccc(C(=O)O)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 2/20 0.35
KDM4E B2RXH2 3/20 0.35
GLA P06280 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DHODH Q02127 3/20 0.34
KDM4C Q9H3R0 4/20 0.34
EGLN1 Q9GZT9 1/20 0.34
KMO O15229 1/20 0.34
TP53 P04637 2/20 0.33
SMURF2 Q9HAU4 1/20 0.33
SMURF1 Q9HCE7 1/20 0.33
NLRP3 Q96P20 1/20 0.33
S1PR1 P21453 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
LMNA P02545 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452936 0.90 NR1H4 (0.35) KMT2ASMN1; SMN2DHODHTP53ALDH1A1
SCHEMBL22452558 0.89 KDM4C (0.42) KDM4EGLAHTTKMT2ASMN1; SMN2
SCHEMBL22453088 0.83 DHODH (0.42) SERPINE1KDM4EGLAHTTKMT2A
SCHEMBL22452822 0.80 DHODH (0.39) KDM4EGLAHTTKMT2ASMN1; SMN2
SCHEMBL22452775 0.78 KDM4E (0.42) KDM4EGLAHTTKMT2ASMN1; SMN2
SCHEMBL22453576 0.78 CYP1A2 (0.40) KDM4EKMT2ASMN1; SMN2KDM4CLMNA
SCHEMBL22453348 0.76 KMT2A (0.42) SERPINE1KDM4EGLAHTTKMT2A
SCHEMBL22453636 0.76 KDM1A (0.40) SERPINE1KMT2ADHODHS1PR1ALDH1A1
SCHEMBL22453296 0.74 HDAC3 (0.47) SERPINE1S1PR1
SCHEMBL22453370 0.71 BACE1 (0.36) ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed