SCHEMBL22453579

SCHEMBL22453579

CCOC(=O)c1cccc(Nc2ccc(N(C)c3ccc(OC(F)(F)F)cc3)cc2C)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
KDM4C Q9H3R0 2/20 0.41
KDM6B O15054 1/20 0.40
MAPT P10636 3/20 0.39
TP53 P04637 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
KDR P35968 2/20 0.38
SCN10A Q9Y5Y9 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LTC4S Q16873 1/20 0.37
AURKA O14965 1/20 0.36
RIPK1 Q13546 1/20 0.36
MLKL Q8NB16 1/20 0.36
RIPK3 Q9Y572 1/20 0.36
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453582 0.90 KDM4C (0.41) CYP1A2KDM4CMAPTTP53MTNR1A
SCHEMBL22453259 0.90 KDM4C (0.44) KDM4CKDM6BKDRSCN10AKDM4E
SCHEMBL22453576 0.81 CYP1A2 (0.40) CYP1A2KDM4CKDM6BMAPTMTNR1A
SCHEMBL22453261 0.80 KDM4C (0.46) KDM4CKDM6BKDM4ENPC1RAB9A
SCHEMBL22453580 0.77 DHODH (0.50) CYP1A2MAPTMTNR1AMTNR1BKDR
SCHEMBL22452936 0.73 NR1H4 (0.35) CYP1A2MAPTTP53SMN1; SMN2
SCHEMBL22452953 0.71 TUBB4A (0.44) CYP1A2KDM4CKDM6BMAPTMTNR1A
SCHEMBL22453458 0.71 MEN1 (0.46) KDM4CKDM6BMAPTPOLBSMN1; SMN2
SCHEMBL18002733 0.70 MAPT (0.46) CYP1A2MAPTSCN10APOLBKDM4E
SCHEMBL31670732 0.68 CYP1A2 (0.66) CYP1A2MAPTPOLBKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed